SYNTHETIC NARCOTIC DRUGS INTRODUCTION
A. General Works
B. Pethidine and Related Compounds
C. Methadone and related compounds
D. Morphinan and morphine synthesis
E. Dithienylbutenylamines and miscellaneous synthetics
Pages: 41 to 47
Creation Date: 1956/01/01
The Bulletin on Narcotics first published a bibliography on synthetic narcotic drugs in Volume III, No. 2, followed by another more comprehensive one in Volume VI, No. 2, and Volume VI, No. 3-4. It is felt, however, that the abundance of new material makes it worthwhile to publish at this time an additional bibliography on the same subject.
This bibliography has no claim to be complete, and information regarding books or articles not included in it would be gratefully received by the Division of Narcotic Drugs, Department of Economic and Social Affairs, European Office of the United Nations, Geneva, Switzerland. As before, this bibliography has been arranged by subject in the following way:
A. General works
B. Pethidine and related compounds
C. Methadone and related compounds
D. Morphinan and morphine synthesis
E. Dithienylbutenylamines and miscellaneous synthetics Under each heading, publications are arranged alphabetically by author. Owing to the nature of the sources available to the secretariat for preparing this bibliography, several titles are given in translation only. They are preceded by an asterisk.
ANONYMUS: Expert Committee on Drugs Liable to Produce Addiction. Fifth report. World Health Organization Technical Report Series, 1955, 95, p 1-16.
BADGER, G. M.; COOK, J. W.; DONALD, G. M. S.; GRAHAM, J. D. P.; WALKER, T.: Synthetic Analgesics . Nature, 1948, 162: 4105, p. 21.
BECKETT, A. H.; CASY, A. F.: Stereochemistry of certain analgesics. Nature, 1954, 173, p. 1231-1232.
-; -: Synthetic analgesics: stereochemical considerations. Journal of Pharmacy and Pharmacology, 1954, 6, p. 986-1001.
BERGEL, F.; MORRISON, A. L.: Synthetic Analgesics, Quarterly Review, 1948, 2: 4, p. 319-382.
BRAENDEN, O. J.; WOLFF, P. O.: Synthetic substances with morphine-like effect. Bulletin of the World Health Organization, 1954, 7: 10, p. 1-25.
DONATELLI, L.: II dolore ed i farmaci antidolorifici (Pain and analgesic drugs). Rassegna Internazionale di Clinica e Terapia, 1955, 35: 1, p. 11-19; ibid. 35: 2, p. 50-59; ibid. 35: 4, p. 128-134.
EISENBERG, W. V.: Microscopic tests for alkaloids and synthetics. Journal of the Association of Official Agricultural Chemists, 1955, 38, p. 653-655.
GADDUM, J. H.: Pharmacology, 4th edition, XVIII + 562 pp. illus. Oxford University Press, New York, 11. (1953).
GEIST, G.: (Addiction dangers of synthetic analgesics). Pharmazeutische Zeitung ver. Apotheker Zeitung, 1953, 89, p. 831-834.
HAAS, H.: (Comparison of analgesics). N. Sch. Archiv für experimentelle Pathologie und Pharmakologie, 1955, 225, p. 442-452.
HILDEBRANDT, F.; MATTHAY, E.: Die Wirkung der starken Analgetica Polamidon, Polamidon C (Polamivet) und Dromoran auf die Darmmotilität. (The effect of powerful analgesics, such as polamidone and polamidone C (polamivet) and dromoran on intestinal motility). N. Sch. Archiv für experimentelle Pathologie und Pharmakologie, 1954, 221: 5, p. 399-403.
KUDAKOVA, N. A.: (Use of non-exchange resins in the determination of pharmaceuticals). Aptechnoe Delo, 1955, 4: 4, p. 34-37.
LESPAGNOL, A.: Les analgésiques centraux de synthèse. Les succédanés synthétiques de l’opium. Actualités pharmacologiques, 1949, 1, p. 145-161; ibid., 1951, 3, p. 27-47.
LEWENSTEIN, Mozels J.: The preparation of compounds having a narcotic effect. British Patent, No. 713675 18 August 1954.
LEWIS, J.R.: A study of the development of tolerance to the actions of 1-Methyl -4-(3-hydroxyphenyl)-4-piperidyl ethyl ketone hydrochloride in dogs. Journal of Pharmacology and Experimental Therapeutics, 1949, 96: 4, p. 410-415.
-; The development of tolerance in rats to some new synthetic analgesics. Journal of Pharmacology and Experimental Therapeutics, 1949, 96: 1, p. 31-37.
LUNDY, J. S.: Development of Analgesia after a century of anesthesia. Journal of the American Medical Association, 1955, 157: 16, p. 1399-1403.
MACDONALD A. D.: Le soulagement de la douleur. Annales Pharmaceutiques Françaises, 1954, 12: 9-10, p. 663-671.
MAROLDA, C. I.: Analgésicos centrales sintéticos (Synthetic central analgesics). Semana Médica, 1955, 106: 11, p. 292-297.
MARTINETTO, G.: (Synthetic analgesics for pre-anesthetic treatment). Minerva Anestesiologica, 1955, 21, p. 86-91.
MERGER, R.; LEVY, J.; BOURRICHON: Effets sur le travail de l'accouchement de l'association analgésique nembutal-dolosal-trilene. Bulletin de la fédération des sociétés de gynécologie et d' obstétrique de langue française, 1953, 5: 3, p. 304-306.
-; MELCHIOR , J.: L'Analgésie obstéricale par l'association médicamenteuse: nembutal-dolosal-trilene. Bulletin de la fédération des sociétés de gynécologie et d'obstétrique de langue française, 1953, 5: 5. p. 301-304.
MILLER, J. W.; ELLIOTT, H. W.: Rat tissue levels of carbon-14 labeled analgetics as related to pharmacological activity. Journal of Pharmacology and Experimental Therapeutics, 1955, 113: 3, p. 283-291.
MORRISON, A. L.; RINDERKNECHT, H.: Synthetic Analgesics. Jubilee Volume Emil Barell (Hoffmann-La Roche), 1946, p. 253-263.
ORTH, O. S.: Newer drugs for general anesthesia. Postgraduate Medicine, 1954, 15: 5, p. 393-398.
PÓRSZÁSZ, J.; KNOLL, J.; KOMLÓS, E.: Wirkung der Parasympathomimetika auf die Analgesie (Effect of parasympathetic substances on analgesia). Acta Physiologica Academiae Scientiarum Hungariae, 1951, 2: 3-4, p. 469-477.
SCHAUMANN, O.: Die Wirkungsspezifität der morphinähnlichen Analgetica (Specificity of action of morphine-like analgetics). Arzneimittel-Forschung, 1954, 4: 3a (special), p. 115-116.
-; (150 years of morphine and 15 years of synthetic morphine-like analgetics). Angewandte Chemie, 1954, 66, p. 765-768.
SOEHRING. K.: Neuere synthetische Arzneimittel mit zentralanalgetischer Wirkung (New synthetic drugs with central analgesic action). Medizinische Klinik, 1950, 45: 27, p. 817-822.
THORP, R. H.: The assessment of analgesic activity in new synthetic drugs. British Journal
.
TSAO, Yer Fang: The preparation of analogs of demerol, amidone, and isoamidone and the reactions of certain nitriles with Grignard reagents. University Microfilms (Ann Arbor, Mich.). Pub. No. 5752, 128 pp.; Dissertations abstracts, 1953, 13: 5, p. 2061.
TSUTOMU, E.: Biochemistry of the poisoning with narcotics. Shizen (Nature), 1954, 9: 5, p. 30-39.
VIDIC, E.; BREINLICH, J.: Zum mikrochemischen Nachweis von Cliradon und Dromoran im Urin (Microchemical determination of cliradon and dromoran in urine). Arzneimittel-Forschung, 1953, 3: 9, p. 490-491.
WALSCH, E. O. F.: Habit-forming drugs and cell metabolism. Pharmaceutical Journal, 1954, 119, p. 483-484.
A
ANDERSEN, H. C.;JEPSEN, O.; KRISTIANSEN, F.: Nystagmus induced by pethidine. Acta Oto-Laryngologica, Supplementum, 1953, 109, p. 9-14.
AREZIO, G.; PERUZZO, L.; VERGA, G.: Azione dei farmaci componenti il cocktail vegetativolitico (cloropromazina, prometazina, mefedina), somministrati isolamente, sul surrene di ratto (Action of the lytic cocktail drugs [chlorpromazine, promethazine, mephedine] administered separately, on the adrenal glands of rats). Acta Anaesthesiologica, 1955, 6: 1, p. 1-10.
ARGENT, D. E.; DINNICK, O. P.: Pethidine phlebitis. British Journal of Anaesthesia, 1954, 26: 4, p. 260-263.
AVISON, A. W. D.; MORRISON, A. L.: Synthetic Analgesics. VI. The synthesis of ketobemidone. Journal of the Chemical Society, 1950, p. 1469-1471. VII. Metadine and related 3-phenyl piperidine derivatives (4304) p. 1471-1474, No. 305. VIII. Further attempts to prepare 3-phenylpiperidine derivatives, p. 1474-1477.
BACHRACH, E. H.; GODHOLM, A. N.; BETCHER, A. M.: Clinical observations on the use of alphaprodine (nisentil) for postoperative analgesia. Surgery, 1955, 37: 3, p. 440-445.
BADGER, G. M; COOK, J. W.; WALKER, T.: Synthesis of Piperidine derivatives. II. Aryldecahydroquinolines. Journal of the Chemical Society, 1948, II, p. 2011-2017.
_____; COOK, J. W.; CROSBIE, G. W.: The chloromethylation of naphtalene and of Tebalin. Journal of the Chemical Society, 1947, II. p. 1432-1434.
BALIAH, V.; GOPALAKRISHNAN, V.: Synthesis of some 4-piperidone derivatives. Journal of the Indian Chemical Society, 1954, 31, p. 250-252.
BARR, W.; COOK, J. W.: Synthesis of Piperidine derivatives, part I. Journal of the Chemical Society, 1945, I. p. 438-441.
BATTERMANN, R. C.: Clinical effectiveness and safety of a new synthetic analgesic drug, Demerol. Archives of International Medicine, 1943, 71: 3, p. 345-356.
-;Demerol; a new synthetic analgesic: its indications as a substitute for morphine. Connecticut Medical Journal, 1944, 8: 1, p. 13-17.
-; MULHOLLAND, J. H.: Demerol; a substitute for morphine in the treatment of postoperative pain. Archives of Surgery, 1943, 46: 3, p. 404-409.
BAZANOVA, S. V.; KLEMENT’EV, F. V.; KISELEVA, K. I.: Sravuitel'noe deistvie atropina, lidola i tifena pri lechenii bol'nykh s of Pharmacology and Chemotherapy, 1946, 1: 2, p. 113-126 diskineticheskimi zaporami (Comparative effects of atropin, lidol and thiphen in Therapy of diskinetic constipation). Sovietskaia Meditsina, 1954, 18: 4, p. 29-31.
BAZANOVA, V. B. S. V.: Promedol-boleuto-liaiushchee sredstbo pr lichenii vnutrennukh zabobevanuy (Promedol-analgesic in the treatment of internal disease). Sovietskaia Meditsina, 1954, 18: 10, p. 39-40.
BELINKOFF, S.: Preoperative sedation with nisentil. Current researches in Anesthesia and Analgesia, 1955, 34: 2, p. 116-118.
BENTHIN, W.: Schmerzlinderung in der Geburt durch Dolantin (Dolantin in delivery). Deutsche Medizinische Wochenschrift, 1940 , 66, p. 760-762.
BERGEL, F.; MORRISON, A. L.; RINDERKNECHT, H.: No. 69 Synthetic Analgesics. II. A new synthesis of Pethidine and similar compounds, p. 265-267; No. 70 III. The action of hydrogen halides on ethers of α α - bis- (B'hydroxyethyl) phenylacetonitrile, p. 267-269. No. 70 IV. Synthesis of 3-substituted piperidino and pyrrolidines, p. 269-272. Journal of the Chemical Society, 1944.
BIEL, J.H.; SPRENGELER, E. P.; LEISER, H. A.; HORNER, J.; DRUKKER, A.; & FRIEDMAN, H. L.: Antispasmodics. II. Derivatives of N-substituted-3-piperidols. Journal of the American Chemical Society, 1955, 77: 8, p. 2250-2256.
BLICKE, F. F.; TSAO, E. P.: Preparation of 1-methyl-4-phenyl-4-(aminomethyl)- and 1-methyl-4-phenyl-4- (methylaminomethyl)-piperidine. Journal of the American Chemical Society, 1953, 75, p. 5417-5418.
BRENDER, H.: Zur Pharmakologie der Phenyl-(1-piperidino) - essigsäure-s - diethylaminoethyl-esters (Pharmacology of 2-(diethylamino-) ethyl phenyl piperidino-acetate). Arzneimittel-For-schung, 1954, 4: 2, p. 67-70.
VON BRUECKE, S.: Ueber Dolantin Abusus und einen Fall von Dolantin delirium (Abuse of dolantin; a case of delirium caused by that drug). Wiener klinische Wochenschrift, 1940, 53, p. 854-856.
BURNS, J. J.; BERGER, B. L.; LIEF, P. A.; WOLLACK, A.; etc.; The physiological disposition and fate of meperidine (demerol) in man and a method for its estimation in plasma. Journal of pharmacology and experimental therapeutics, 1955, 114: 3, p. 289-298.
CALZOLARI, G.: Analgesia profonda ed anestesia locale nella chirurgia della tiroide (Deep analgesia and local anesthesia in thyroid surgery). Minerva anestesiologica, 1955, 21: 6, p. 141-143.
CLARK, B. B.: The effect of syntropan, demerol, and trasentine on gastric secretion. Federation Proceedings, 1947, 6: 1, Part I, p. 48.
CLIMENKO, D. R.: Demerol: A pharmacologically active substance with atropine-like and morphine-like properties. Federation Proceedings, 1942, 1, p. 15.
COLLADOS STORNI, M. P.: Anestesia con petidina endovenosa para amigdalectomias; comunication prevista (Pethidine intravenous anesthesia in tonsillectomy; preliminary communication). Revista de la Facultad de ciencias médicas de la Universidad nacional de Cordoba, 1953, 11: 3-6, p. 627-631.
COMINSKY, N. C.: The effect of demero and morphine on the histologic: tructure of mouse tissues. Texas Reports on Biology an d Medicine, 1955, 13: 2, p. 222-233.
COOK, A. H.; REED, K.J.: No. 98: Experiments in the piperidine series. Journal of the Chemical Society, 1945, I, p. 399-402.
COSTA, P. J.; BONNYCASTLE, D. D.: The effect of levallorphan tartrate, nalorphine HCl and WIN 7681 (l-allyl-4-phenyl-4-carbethoxy-piperidin), on respiratory depression and analgesia induced by some active analgetics. Journal of Pharmacology and Experimental Therapeutics, 1955, 113: 3, p. 310-318.
CRIMENI, R.: Osservazioni cliniche sull'azione pre-anestetica del cliradon (Clinical observations on the pre-anesthetic effects of cliradon). Gazzetta medica italiana, 1953, 112: 8, p. 203-206.
CRIPPS, J. A. R.; HALL, B.; HAULTAIN, W. F. T.: Analgesia in labour; record of 102 cases treated with pethidine. British Medical Journal, 1944, No. 4371, p. 498-500.
DEXEUS TRIAS DE BES J. M.; SEGUR FERRER, J. M.: La associación largactil-dolantina-pituitrina en la conduccion del parto. (Combined largactil, dolantin and pituitrin in management of labour). Revista Española de Obstetrica y Ginecologia, 1955, 14: 81, p. 132-137
DIETRICH, H.: Klinische Erfahrungen mit einem neuen synthetischen Spasmolyticum und Analgeticum (Clinical experiments with a new synthetic analgesic). - Deutsche medizinische Wochenschrift, 1939, 65, p. 969-970.
EIDINOVA, M. B.: Primenenie promedola pri zabolevaniakh nervnoi sistemi (Use of promedol in diseases of the nervous system). Sovietskaia meditsina, 1954, 18: 11, p. 12-14.
ELLIOTT, H. W.: Comparative effects of 1,1- diphenyl-l-(dimethylamino -isopropyl)- bu-temone-2 (10820) demerol and morphine on the respiration of rat cerebral cortex slices. Federation Proceedings, 1947, 6 Part II, p 327-328.
ERLENDSSON, V.: Dolantin "Bayer ". Ugeskrift for Laeger, 1940, 102; p. 1330-1331.
FEHER, V.; BRUTAR, V.: Uziti dolsinu pri porodu (Use of dolsin in labour). Ceskoslovenska gynaekologie,1953, 18 : 4, p. 360-372.
FERRER, M. L.; SOKOLOFF, L.: The antidiuretic effect of morphine and Demerol in congestive heart failure. American Journal of medical science,1947, 214 : 4, p. 372-384.
FERRON, M.: Nisentil; analgésique obstétrical. Union Médicale du Canada,1955, 84 : 4, p. 431-433.
FINKELSTEIN, J.; LEE, J.: Piperidine derivatives. U. S. Patent No. 2,686,784, 17 August 1954 (Hoffmann-La Roche Inc.).
FITZGERALD, G.; McARDLE, B.: Effect of pethidine on pain in neurological cases. Lancet,1943, No. 6236, p. 296-297.
FORTI, D.: Procaina e dolantinici per via endovenosa in anestesia ed analgesia postoperatoria (Intraveinous procaine and dolantinin anesthesia and postoperative analgesia). Minerva Anestesiologica,1953, 19 : 8, p. 216-217.
FOSTER, R. H. L.; CARMAN, A. J.: Studies in analgesia: piperidine derivatives with morphine-like activities. Journal of Pharmacology and Experimental Therapeutics,1949, 91 : 3, p. 195-209.
FROMMEL, E.; RADOUCO-THOMAS, C.: De l'incidence des ganglioplégiques sur la prépararion de la narcose au pentothal par la morphine et le dolosal; du danger des opiacés. Praxis,1955, 44 : 18, p. 407-409.
GALLEN. B.; PRESCOTT, F.: Pethidine as an obstetric analgesic-a report on 150 cases. British Medical Journal,1944, No. 4335, p. 176-179.
GAMMELTOFT, A.; JOHANSEN, S. H.; RUBEN, H.: Pethidin ved cystoskopi; erfaringer med pethidin intravenost ved endoskopi af urethra og blaere hos maend (Pethidine in cystoscopy; experience with intravenous pethidine in endoscopy of male urethra and bladder). Ugeskrift for Laeger,1 953, 115 : 39, p. 1448-1449.
----------------; Intravenous pethidine for oesophagoscopy and gastroscopy. Anaesthesia,1953, 8 : 3, p. 194.
GEFTER, A. I.; MATUSOVA, A. P.: Primenenie tifen-promedola pri koronarnoi bolezni (Use of tiphen-promedol in coronary disease). Sovietskaia Meditsina,1955, 19 : 8, p. 22-25.
GLAZEBROOK, A. J.; BRANWOOD, A. W.: Clinical trials of β-pethidine. Lancet,1945, 249 : 6374, p. 528-529.
GORDON, G. S.; DIXON, A. B.: Observations on Demerol as an obstetric analgesic. American Journal of Obstetrics and Gynecology,1943, 45,p. 320.
GREBENNIK, L. I.: (Elimination of promedol from the body). Farmakologiya Toksikologiya,1954, 17 : 4, p. 48-51.
GYERMEK, L.: Studies on cholinergic blocking substances. VIII. Pharmacological actions of certain polymethylene-, bis- and azapentylenebis-pyrrolidine and piperidine derivatives. Acta Physiologica Academiae Scientiarum Hungaricae,1955, 8 : 1, p. 49-60.
HALLE, J.; DECHENE, J. P,; MONTMINY, L.; PARADIS, G.: Le nisentil en bronchoscopie. Laval médical,1955, 20:1, p. 5256.
HARDY, J. D.; McKEEN CATTELL: Measurement of pain threshold raising action of aspirin, codeine and meperidine (Demerol). Federation Proceedings,1950, 9 : 1, Part I, p. 282.
HARVEY, W. P.; BERKMAN, F.; LEONARD, J.: Caution against the use of meperidine hydrochloride (isonipecaine, demerol) in patients with heart disease, particularly auricular flutter. American Heart Journal,1955, 49 : 5, p. 758-769.
HECHT, H.; NOTH, P. H.; YONKMAN, F. F.: Demerol; clinical observations. Journal of the American Medical Association,1943, 121 : 16, p. 1307.
HEIDT, T. J.; DALLIS, N. P.; O'CONNELL, W.J.: The use of Demerol in artificial fever. American Journal of Psychiatry,1945, 101 : 6,p. 789-792.
HERSCHFUS, J. A.; SALOMON, A.; SEGAL, M. S.: The use of demerol in patients with bronchial asthma. Annals of Internal Medicine,1954, 40 : 3, p. 506-515.
HOCH, D.; KARRER, P.: Synthèse de plusieurs homologues de la methyl-piperidine. Helvetica Chimica Acta,1954, 37,p. 397-402.
HORÁKOVÉ, Z.; VOTAVA, Z.: Analgetické účinek morfinu, dolsinu a mecodinu pri ruznem zpusobu podání farmakologické studie (Analgetic effect of morphine, dolsin and mecodin in various ways of application; a pharmacological study). Ceskoslovenské Farmacie,1955, 4: 3, p. 131-133.
HURLBUT, D. B.; D1LLE, J. M.: The effect of nisentil upon the intra-uterine respiratory movements of the rabbit fetus. Anesthesiology,1952, 13 : 1, p. 71-76.
----------------; ----------------: The effect of nisentil upon the intra-uterine respiratory movements of the rabbit fetus. Journal of Pharmacology and Experimental Therapeutics,1951, 103:4, p. 348.
IZAR, G.; IENZI, S.: Studi sulla Dolantina. (Study on Dolantine). Rassegna internaz, di clinica e terapia,1941, 22,p. 213-221, 251-256.
JENSEN, K. A.; LUNDQUIST, F.; REKLING; WOLFFBRANDT, C. A.: Ein neuer Typus von Piperidin Derivaten mit analgeter und spasmolyter Wirkung (A new type of piperidine-derivative with analgesic and spasmolytic activity). Chemisches Zentralblatt,1944, I. 115 : 5, p. 297-298.
JESSEN, H.: Dolantin in recurrent hiccups. Journal of the American Medical Association,1942, 118:8, p. 674-675.
-;Om Dolantin. Ugeskrifi for Laeger,1940, 102,p. 1326-1328.
KLEIN, E. K.: Erfahrungen mit Dolantin, einem myotrop und neurotrop wirkenden Spasmolytikum (Experience with Dolantin, a Spasmolytic working as myotrop and neuro-trop). Münchener medizinische Wochenschrift,1939 2, p. 1676.
KRACHEEL,E.: Die Leistungsfähigkeit der Blutnarkose, ein Beitrag zum Narkoseproblem der chirurgischen Praxis (Potentiation of intraveinons anesthesia, a contribution to the anesthesia problem of surgical practice). Zentralblatt für Chirurgie,1955, 80 : 10, p. 398-405.
KUCHER, I.: Zwei Fälle von Dolantinsucht. (Two cases of addiction to dolantin). Klinische Wochenschrift,1940, 19;p. 688-489.
KUNZ, T.: Die Dolantin-Evipan-Lachgas-narkose mit My 301 als Muskelrelaxans (Dolantin-evipan nitrous oxide anesthesia with My 301 as a muscle relaxant). Medizinische,1953, No. 48, p. 1555-1556.
KWARTLER, C. F.: U.S. patent No. 2,634,275, 7 April 1953. 4-acylamino-l-alkyl-4-phenyl-piperidines and method of making same.
LAGARDE, L. A.; ORTIZ DE LA PENA, R.; BRAVO SERRADELL, O.: Tres drogas auxiliares en obstetricia (Three auxiliary drugs in obstetrics). Ginecologia y Obstetricia de Mexico,1955, 10 : 2, p. 140-150.
LEE, J.; ZIERING, A.; BERGER, L.; HEINEMAN, S. D.: Studies on the synthesis of Analgesic compounds. Jubilee Volume Emil Barell,(Hoffmann-La Roche), 1946, p. 265-305.
LEWIS, J. R.: Action of l-methyl-4-(3-Hydroxy phenyl)-4-piperidyl ethyl ketone on the gastrointestinal tract. Proceedings of the Society for Experimental Biology and Medicine,1949, 71: 2,p. 300-303.
McELVAIN, S. M.; DICKINSON, W. B.; ATHEY, R.: Piperidine derivatives XXV. Reaction of certain 3-substitutes l-methyl-4-piperidones with organometallic compounds. Journal of the American Chemical Society,1954, 76, p. 5625-5633.
----------------; BERGER, R. S.: Piperidine derivatives. XXVII. The condensation of 4-piperidones and piperidinols with phenols. Journal of the American Chemical Society,1955, 77:10, p. 2848-2850.
MARTIN, C.: L'anesthésie de base diparcoldolosal en chirurgie gériatrique et chez le malade représentant un manvais risque. Anes-thésie et Analgésie,1955, 12: 2, p. 335-347.
Motatovo MATSUMOTO; Yasumichi KISHINOUXE; Iwao YAMAZAKI; Yoshio NAKAMURA: Synthesis of N-ethylpiperldine. Coal Tar,1954, 6, p. 198-201.
MOREL-FATIO, D.: A propos de 200 cas d'anesthésie de base (diparcol-dolosal)+ locale en chirurgie réparatrice. Anesthésie et Analg?ie,1955, 12 : 2, p. 348-357.
MORISOT, D.: L'association diehazine-p?hidine I. V. (dipdol) comme anesth?ie de base. Anesthésie et Analgésie,1955, 12:2, p. 365-368.
NAZAROV, Z. N.; NOKOLOV, D. V.; RAKCHEEVA, V. N.: Geterotsiklicheskie soedinenu?ia. XXX. Stereoizomeriia 2, 5-di-metil-4-piperidola, 1, 2, 5-trimetil-4-piperidola i ikh proizvodnykh (Heterocyclic compounds. XXIX. Stereoisomers of 2, 5-dimethyl-4-piperidol, 1, 2, 5-trimethyl-4-piperidol and their derivatives). Izvestia Akademii Nauk SSSR otdelenie Khissicheskikh Nauk,1954, No. 1, p. 80-94.
NICKERSON, M.; GOODMAN, L. S.: Synergistic isonipeca ?ne-amphetamine analgesia. Federatiuo Proceedings,1947, 6 : 1, part II p. 360.
ORKIN, L. R.; EGGE, R. K., ROVENSTINE, E. A.: Effect of nisentil, meperidine and morphine on respiration in man. Anesthesiology,1955, 16: 5, p. 699-707.
PASSMORE, G. G.; SANTA CRUZ, E. W.: The use of intravenous and intramuscular injections of demerol and scopolamine in labor and delivery. American Journal of Obstetrics and Gynecology, 1954, 68 : 4, p. 998-1008.
PATERSON, S. J.; PRESCOTT, F.: Nalorphine in the prevention of neonatal asphyxia due to maternal sedation with pethidine. Lancet,1954, 266 : 6810, p. 490-493.
PERRINE, T. D.; MAY, E. L.: Synthesis of 6-dimethylamino-4, 4-diphenyl-heptane and other compounds related to Demerol. Journal of Organic Chemistry, 1954, 19,p. 773-779.
PÓRSZÁSZ, J.; VENULET, .J.; GIBSZER PÓRSZÁSZ , K.: Untersuchungen über die Synergisierbarkeit der Analgetika; Wirkung des Doryls und Physostigmins auf die Verteilung'des Dolantins im Organisnms (Studies on synergism of analgesics; effect of doryl and physostigmine on the distribution of dolantin in the organism). Acta physiologica academiae scientiarum hungaricae, 1954, 5 : 3-4, p. 509-519.
PRESTON, F. S.: Anaesthesia for mitral valvotomy. British Journal of anaesthesia, 1953, 25 : 4, p. 299-314.
PRYOR, W. J.: Pethidine in anesthesia. New Zealand Medical Journal, 1953, 52 : 291, p. 398-400.
RANDALL, L. O.; LEHMANN, G.: Pharmacological studies on analgesic piperidine derivatives. Journal of Pharmacology and Experimental Therapeutics, 1948, 93 : 3, p. 314-328.
RASOR, R. W.; CRECRAFT, H. J.: Addiction to Meperidine (Demerol) hydrochloride. Journal of the American Medical Association, 1955, 157 : 8, p. 654-657.
REISINGER, F.: Das neue Analgeticum und Spasmolyticum Dolantin (A new analgesic and spasmolytic; dolantin). Wiener medizinische Wochenschrift, 1940, 90,p. 400.
ROBERTS, H.; WRIGLEY, F.: Nisentil in obstetrics; clinical trials with a new analgesic. Journal of Obstetrics and Gynaecology of the British Empire, 1953, 60 : 4, p. 538-540.
ROBY, C.; SCHUMANN, W. R.; Demerol (S-140) and scopolamine in labor: a preliminary report. American Journal of Obstetrics and Gynecology, 1943, 45,p. 318.
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COUNCIL on pharmacy and chemistry : New and unofficial remedies: levorphane tartrate. Journal of the American medical association, 1954, 156 : 3, p. 250-251.
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